PHA767491 HCl抑制劑PHA-767491 is an effective ATP-competitive dual Cdc7/CDK9 inhibitor (IC50: 10/34 nM). It has ~20-fold selectivity against GSK3-β and CDK1/2, 50-fold selectivity against CDK5 and MK2, 100-fold selectivity against CHK2 and PLK1.
產(chǎn)品名稱: | PHA767491 HCl | ||
英文名: | PHA767491 HCl | ||
CAS NO.: | 942425-68-5 | ||
分子式: | C12H12ClN3O | ||
分子量: | 249.696181297302 | ||
產(chǎn)品品牌: | targetmol | ||
產(chǎn)品規(guī)格: | 2mg |